The one-pot synthesis of amidonapthoquinones from aminonaphthoquinones
نویسندگان
چکیده
منابع مشابه
A laccase-catalysed one-pot synthesis of aminonaphthoquinones and their anticancer activity.
Nuclear monoamination of a 1,4-naphthohydroquinone with primary aromatic amines was catalysed by the commercial laccase, Novozym 51003, from Novozymes to afford aminonaphthoquinones. The synthesis was accomplished by reacting a mixture of the primary amine and 1,4-naphthohydroquinone in succinate-lactate buffer and a co-solvent, dimethylformamide, under mild reaction conditions in a vessel open...
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ژورنال
عنوان ژورنال: Tetrahedron Letters
سال: 2020
ISSN: 0040-4039
DOI: 10.1016/j.tetlet.2020.151800